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Cetrorelix diacetate
CAS No. 130143-01-0
Cetrorelix diacetate ( SB-75 diacetate )
产品货号. M21741 CAS No. 130143-01-0
Cetrorelix diacetate (SB-075 diacetate) 是一种有效的促性腺激素释放激素 (GnRH) 受体拮抗剂，IC50 为 1.21 nM。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥745 | 有现货 |
|
| 10MG | ￥1239 | 有现货 |
|
| 25MG | ￥2487 | 有现货 |
|
| 50MG | ￥3726 | 有现货 |
|
| 100MG | ￥5476 | 有现货 |
|
| 500MG | ￥11583 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Cetrorelix diacetate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Cetrorelix diacetate (SB-075 diacetate) 是一种有效的促性腺激素释放激素 (GnRH) 受体拮抗剂，IC50 为 1.21 nM。
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产品描述Cetrorelix diacetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix diacetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.(In Vitro):Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
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体外实验Cetrorelix diacetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix diacetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
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体内实验——
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同义词SB-75 diacetate
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通路GPCR/G Protein
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靶点Other Targets
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number130143-01-0
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分子量1551.14
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分子式C??H???ClN??O??
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纯度>98% (HPLC)
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溶解度——
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SMILES——
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化学全称Ac-{2-Naph-Ala}-{Cl-Phe}-{3Py-Ala}-SY-{Cit}-LRPA-NH2
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Beckers T et al. Characterization of gonadotropin-releasing hormone analogs based on a sensitive cellular luciferase reporter gene assay. Anal Biochem. 1997 Aug 15;251(1):17-23.
2. Gründker C et al. Role of gonadotropin-releasing hormone (GnRH) in ovarian cancer. Reprod Biol Endocrinol. 2003 Oct 7;1:65.
产品手册
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Cetrorelix diacetate
Cetrorelix diacetate (SB-075 diacetate) 是一种有效的促性腺激素释放激素 (GnRH) 受体拮抗剂，IC50 为 1.21 nM。
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